The first potent inhibitor of mammalian group X secreted phospholipase A2: elucidation of sites for enhanced binding.
第一作者:
Brian P,Smart
第一单位:
Department of Chemistry and Biochemistry, University of Washington, Seattle, Washington 98195, USA.
作者:
主题词
动物(Animals);结合部位(Binding Sites);结晶学, X线(Crystallography, X-Ray);Ⅹ型磷脂酶A2(Group X Phospholipases A2);人类(Humans);吲哚类(Indoles);小鼠(Mice);模型, 分子(Models, Molecular);磷脂酶A(Phospholipases A);磷脂酶类A2(Phospholipases A2);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm060136t
PMID
16686528
发布时间
2025-05-29
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