High content screening identifies decaprenyl-phosphoribose 2' epimerase as a target for intracellular antimycobacterial inhibitors.
第一作者:
Thierry,Christophe
第一单位:
Screening Technologies and Pharmacology, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea.
作者:
主题词
动物(Animals);抗生素类, 抗结核(Antibiotics, Antitubercular);苯甲酰胺类(Benzamides);细胞生长过程(Cell Growth Processes);细胞, 培养的(Cells, Cultured);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物发现(Drug Discovery);人类(Humans);巨噬细胞(Macrophages);小鼠(Mice);微生物敏感性试验(Microbial Sensitivity Tests);显微镜检查, 共焦(Microscopy, Confocal);显微镜检查, 荧光(Microscopy, Fluorescence);结核分枝杆菌(Mycobacterium tuberculosis);主成分分析(Principal Component Analysis);消旋酶类和差向异构酶类(Racemases and Epimerases);结果可重复性(Reproducibility of Results);构效关系(Structure-Activity Relationship);结核(Tuberculosis)
DOI
10.1371/journal.ppat.1000645
PMID
19876393
发布时间
2022-03-10
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PLoS pathogens
e1000645页
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