2005年第67卷05期
共45篇1. Palmitoylation of the 5-hydroxytryptamine4a receptor regulates receptor phosphorylation, desensitization, and beta-arrestin-mediated endocytosis. 1434-43页
作者:Evgeni,Ponimaskin; Aline,Dumuis; Florence,Gaven; Gaël,Barthet; Martin,Heine; Konstantin,Glebov; Diethelm W,Richter; Martin,Oppermann
2. Constitutive activation and environmental chemical induction of the aryl hydrocarbon receptor/transcription factor in activated human B lymphocytes. 1740-50页
作者:Lenka L,Allan; David H,Sherr
3. The effect of hydroxylamine on KATP channels in vascular smooth muscle and underlying mechanisms. 1723-31页
作者:Guanghua,Tang; Lingyun,Wu; Rui,Wang
4. Aspects of dioxin toxicity are mediated by interleukin 1-like cytokines. 1393-8页
作者:Kalyan,Pande; Susan M,Moran; Christopher A,Bradfield
5. Amino acids critical for substrate affinity of rat organic cation transporter 1 line the substrate binding region in a model derived from the tertiary structure of lactose permease. 1600-11页
作者:Christian,Popp; Valentin,Gorboulev; Thomas D,Müller; Dmitry,Gorbunov; Natalia,Shatskaya; Hermann,Koepsell
6. Effect of azelnidipine on angiotensin II-mediated growth-promoting signaling in vascular smooth muscle cells. 1666-73页
作者:Jian-Mei,Li; Masaru,Iwai; Tai-Xing,Cui; Li-Juan,Min; Masahiro,Tsuda; Jun,Iwanami; Jun,Suzuki; Masaki,Mogi; Masatsugu,Horiuchi
7. Long-term nicotine treatment decreases striatal alpha 6* nicotinic acetylcholine receptor sites and function in mice. 1639-47页
作者:Albert,Lai; Neeraja,Parameswaran; Mirium,Khwaja; Paul,Whiteaker; Jon M,Lindstrom; Hong,Fan; J Michael,McIntosh; Sharon R,Grady; Maryka,Quik
8. Heparan sulfate regulates the antiangiogenic activity of endothelial monocyte-activating polypeptide-II at acidic pH. 1534-43页
作者:Sun-Young,Chang; Hyun-Jeong,Ko; Tae-Hwe,Heo; Chang-Yuil,Kang
9. Mechanism of the anti-inflammatory effect of thiazolidinediones: relationship with the glucocorticoid pathway. 1620-8页
作者:Armando,Ialenti; Gianluca,Grassia; Paola,Di Meglio; Pasquale,Maffia; Massimo,Di Rosa; Angela,Ianaro
10. Beta-adrenergic receptor stimulation promotes G alpha s internalization through lipid rafts: a study in living cells. 1493-504页
作者:John A,Allen; Jiang Z,Yu; Robert J,Donati; Mark M,Rasenick
11. Cephalostatin 1 inactivates Bcl-2 by hyperphosphorylation independent of M-phase arrest and DNA damage. 1684-9页
作者:Irina M,Müller; Verena M,Dirsch; Anita,Rudy; Nancy,López-Antón; George R,Pettit; Angelika M,Vollmar
12. Superagonistic action of 14-epi-analogs of 1,25-dihydroxyvitamin D explained by vitamin D receptor-coactivator interaction. 1566-73页
作者:Guy,Eelen; Lieve,Verlinden; Natacha,Rochel; Frank,Claessens; Pierre,De Clercq; Maurits,Vandewalle; Giuseppe,Tocchini-Valentini; Dino,Moras; Roger,Bouillon; Annemieke,Verstuyf
13. Subtype-specific affinity for corticosterone of rat organic cation transporters rOCT1 and rOCT2 depends on three amino acids within the substrate binding region. 1612-9页
作者:Valentin,Gorboulev; Natalia,Shatskaya; Christopher,Volk; Hermann,Koepsell
14. The breast cancer resistance protein (BCRP/ABCG2) affects pharmacokinetics, hepatobiliary excretion, and milk secretion of the antibiotic nitrofurantoin. 1758-64页
作者:Gracia,Merino; Johan W,Jonker; Els,Wagenaar; Antonius E,van Herwaarden; Alfred H,Schinkel
15. The human organic anion transporter 2 gene is transactivated by hepatocyte nuclear factor-4 alpha and suppressed by bile acids. 1629-38页
作者:Katrin,Popowski; Jyrki J,Eloranta; Michael,Saborowski; Michael,Fried; Peter J,Meier; Gerd A,Kullak-Ublick
16. Investigations of calsequestrin as a target for anthracyclines: comparison of functional effects of daunorubicin, daunorubicinol, and trifluoperazine. 1505-12页
作者:Henry A,Charlier; Richard D,Olson; Carissa M,Thornock; Wendy K,Mercer; David R,Olson; T Stephen,Broyles; Dawn J,Muhlestein; Corianton L,Larson; Barry J,Cusack; Susan E,Shadle
17. A novel and efficient approach to discriminate between pre- and post-transcription HIV inhibitors. 1574-80页
作者:Dirk,Daelemans; Christophe,Pannecouque; George N,Pavlakis; Oriana,Tabarrini; Erik,De Clercq
18. A synthetic derivative of the natural product rocaglaol is a potent inhibitor of cytokine-mediated signaling and shows neuroprotective activity in vitro and in animal models of Parkinson's disease and traumatic brain injury. 1544-55页
作者:T,Fahrig; I,Gerlach; E,Horváth
19. Transcriptional regulation of mouse mu opioid receptor gene: Sp3 isoforms (M1, M2) function as repressors in neuronal cells to regulate the mu opioid receptor gene. 1674-83页
作者:Hack Sun,Choi; Cheol Kyu,Hwang; Chun Sung,Kim; Kyu Young,Song; Ping-Yee,Law; Li-Na,Wei; Horace H,Loh
20. Adenosine A2A receptor stimulation increases angiogenesis by down-regulating production of the antiangiogenic matrix protein thrombospondin 1. 1406-13页
作者:Avani,Desai; Cassandre,Victor-Vega; Swathi,Gadangi; M Carmen,Montesinos; Charles C,Chu; Bruce N,Cronstein
21. Differential modulation of glutamatergic transmission by 3,5-dibromo-L-phenylalanine. 1648-54页
作者:V,Yarotskyy; A V,Glushakov; C,Sumners; N,Gravenstein; D M,Dennis; C N,Seubert; A E,Martynyuk
22. Vacuolar degradation of rat liver CYP2B1 in Saccharomyces cerevisiae: further validation of the yeast model and structural implications for the degradation of mammalian endoplasmic reticulum P450 proteins. 1460-9页
作者:Mingxiang,Liao; Victor G,Zgoda; Bernard P,Murray; Maria Almira,Correia
23. Structural features of the glutamate binding site in recombinant NR1/NR2A N-methyl-D-aspartate receptors determined by site-directed mutagenesis and molecular modeling. 1470-84页
作者:Philip E,Chen; Matthew T,Geballe; Phillip J,Stansfeld; Alexander R,Johnston; Hongjie,Yuan; Amanda L,Jacob; James P,Snyder; Stephen F,Traynelis; David J A,Wyllie
24. Alpha 2-adrenergic agonist enrichment of spinophilin at the cell surface involves beta gamma subunits of Gi proteins and is preferentially induced by the alpha 2A-subtype. 1690-6页
作者:Ashley E,Brady; Qin,Wang; Patrick B,Allen; Mark,Rizzo; Paul,Greengard; Lee E,Limbird
25. The aminosteroid phospholipase C antagonist U-73122 (1-[6-[[17-beta-3-methoxyestra-1,3,5(10)-trien-17-yl]amino]hexyl]-1H-pyrrole-2,5-dione) potently inhibits human 5-lipoxygenase in vivo and in vitro. 1751-7页
作者:Christian,Feisst; Dana,Albert; Dieter,Steinhilber; Oliver,Werz
26. Identification and characterization of a functional TATA box polymorphism of the UDP glucuronosyltransferase 1A7 gene. 1732-9页
作者:Tim O,Lankisch; Arndt,Vogel; Stefan,Eilermann; Anette,Fiebeler; Britta,Krone; Ayse,Barut; Michael P,Manns; Christian P,Strassburg
27. Pharmacological discrimination of calcitonin receptor: receptor activity-modifying protein complexes. 1655-65页
作者:Debbie L,Hay; George,Christopoulos; Arthur,Christopoulos; David R,Poyner; Patrick M,Sexton
28. Internal PDZ ligands: novel endocytic recycling motifs for G protein-coupled receptors. 1388-90页
作者:JoAnn,Trejo
30. Sex-dependent expression and activity of the ATP-binding cassette transporter breast cancer resistance protein (BCRP/ABCG2) in liver. 1765-71页
作者:Gracia,Merino; Antonius E,van Herwaarden; Els,Wagenaar; Johan W,Jonker; Alfred H,Schinkel
32. Concurrent stimulation of cannabinoid CB1 and dopamine D2 receptors enhances heterodimer formation: a mechanism for receptor cross-talk? 1697-704页
作者:Christopher S,Kearn; Katherine,Blake-Palmer; Emma,Daniel; Ken,Mackie; Michelle,Glass
33. Marked depletion of glycosylation sites in HIV-1 gp120 under selection pressure by the mannose-specific plant lectins of Hippeastrum hybrid and Galanthus nivalis. 1556-65页
作者:Jan,Balzarini; Kristel,Van Laethem; Sigrid,Hatse; Matheus,Froeyen; Els,Van Damme; Anders,Bolmstedt; Willy,Peumans; Erik,De Clercq; Dominique,Schols
35. Antiangiogenic and vascular-targeting activity of the microtubule-destabilizing trans-resveratrol derivative 3,5,4'-trimethoxystilbene. 1451-9页
作者:Mirella,Belleri; Domenico,Ribatti; Stefania,Nicoli; Franco,Cotelli; Luca,Forti; Vanio,Vannini; Lucia Anna,Stivala; Marco,Presta
36. Potentiation of P2Y receptors by physiological elevations of extracellular K+ via a mechanism independent of Ca2+ influx. 1705-13页
作者:Samantha J,Pitt; Juan,Martinez-Pinna; Eric A,Barnard; Martyn P,Mahaut-Smith
37. The general anesthetic isoflurane depresses synaptic vesicle exocytosis. 1591-9页
作者:Hugh C,Hemmings; Wayne,Yan; Robert I,Westphalen; Timothy A,Ryan
38. Developmental regulation of beta-carboline-induced inhibition of glycine-evoked responses depends on glycine receptor beta subunit expression. 1783-96页
作者:Jean-Marie,Mangin; Laurent,Nguyen; Catherine,Gougnard; Grégory,Hans; Bernard,Rogister; Shibeshih,Belachew; Gustave,Moonen; Pascal,Legendre; Jean-Michel,Rigo
40. Effects of valproic acid derivatives on inositol trisphosphate depletion, teratogenicity, glycogen synthase kinase-3beta inhibition, and viral replication: a screening approach for new bipolar disorder drugs derived from the valproic acid core structure. 1426-33页
作者:B J,Eickholt; G J,Towers; W J,Ryves; D,Eikel; K,Adley; L M J,Ylinen; N H,Chadborn; A J,Harwood; H,Nau; R S B,Williams
41. The repertoire of G-protein-coupled receptors in fully sequenced genomes. 1414-25页
作者:Robert,Fredriksson; Helgi B,Schiöth
42. Subtype-specific sorting of the ETA endothelin receptor by a novel endocytic recycling signal for G protein-coupled receptors. 1581-90页
作者:Joachim D,Paasche; Toril,Attramadal; Kurt,Kristiansen; Morten P,Oksvold; Heidi K,Johansen; Henrik S,Huitfeldt; Svein G,Dahl; Håvard,Attramadal
43. U937 cell necrosis mediated by peroxynitrite is not caused by depletion of ATP and is prevented by arachidonate via an ATP-dependent mechanism. 1399-405页
作者:Orazio,Cantoni; Andrea,Guidarelli; Letizia,Palomba; Mara,Fiorani
44. A natural CYP2B6 TATA box polymorphism (-82T--> C) leading to enhanced transcription and relocation of the transcriptional start site. 1772-82页
作者:Jörg,Zukunft; Thomas,Lang; Tanja,Richter; Karen I,Hirsch-Ernst; Andreas K,Nussler; Kathrin,Klein; Matthias,Schwab; Michel,Eichelbaum; Ulrich M,Zanger