Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanones.
第一作者:
Thomas,Beckers
第一单位:
Department of Pharmaceutical Chemistry I, University of Regensburg, D-93040 Regensburg, Germany.
作者:
医学主题词
抗肿瘤药(Antineoplastic Agents);细胞系, 肿瘤(Cell Line, Tumor);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);吲哚类(Indoles);磷酰化(Phosphorylation);嘧啶类(Pyrimidines);喹唑啉类(Quinazolines);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmc.2011.11.023
PMID
22169601
发布时间
2018-12-01
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