Abrogation of the selectivity of adriamycin for negatively-charged phospholipids by 14-valerate side chain substitution.
第一作者:
T G,Burke
第一单位:
Department of Medical Oncology and Therapeutics Research, City of Hope National Medical Center, Duarte, CA 91010-0269.
作者:
主题词
抗生素类, 抗肿瘤(Antibiotics, Antineoplastic);心磷脂质类(Cardiolipins);化学现象(Chemical Phenomena);化学, 物理(Chemistry, Physical);二肉豆蔻磷脂酰胆碱(Dimyristoylphosphatidylcholine);多柔比星(Doxorubicin);动力学(Kinetics);脂双层(Lipid Bilayers);膜, 人工(Membranes, Artificial);容积渗克分子浓度(Osmolar Concentration);磷脂酰甘油类(Phosphatidylglycerols);磷脂类(Phospholipids);构效关系(Structure-Activity Relationship)
PMID
2383860
发布时间
2016-11-23
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