Novel 2,4-diamino-5-substituted-pyrrolo[2,3-d]pyrimidines as classical and nonclassical antifolate inhibitors of dihydrofolate reductases.
第一作者:
A,Gangjee
第一单位:
Division of Medicinal Chemistry, Graduate School of Pharmaceutical Sciences, Duquesne University, Pittsburgh, Pennsylvania 15282, USA.
作者:
医学主题词
叶酸拮抗剂(Folic Acid Antagonists);人类(Humans);肽合酶类(Peptide Synthases);嘧啶类(Pyrimidines);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1021/jm00012a016
PMID
7783147
发布时间
2019-07-09
基金项目
AI30900/AI/NIAID NIH HHS/United States
CA43500/CA/NCI NIH HHS/United States
GM40998/GM/NIGMS NIH HHS/United States
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