Synthesis and quantitative structure-activity relationships of N-(1-benzylpiperidin-4-yl)phenylacetamides and related analogues as potent and selective sigma1 receptor ligands.
第一作者:
Y,Huang
第一单位:
Department of Radiology-PET Center, Wake Forest University School of Medicine, Winston-Salem, North Carolina 27157, USA.
作者:
医学主题词
乙酰胺类(Acetamides);乙酰苯胺类(Acetanilides);动物(Animals);苯甲酰胺类(Benzamides);脑(Brain);豚鼠(Guinea Pigs);配体(Ligands);肝(Liver);男(雄)性(Male);哌啶类(Piperidines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 多巴胺D2(Receptors, Dopamine D2);受体, Σ(Receptors, sigma);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm980032l
PMID
9632369
发布时间
2007-11-14
基金项目
DA 09142/DA/NIDA NIH HHS/United States
NS 33742/NS/NINDS NIH HHS/United States
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