Use of the nitrile oxide cycloaddition (NOC) reaction for molecular probe generation: A new class of enzyme selective histone deacetylase inhibitors (HDACIs) showing picomolar activity at HDAC6
作者:
Kozikowski AP [1]
;
Tapadar S [2]
;
Luchini DN ;
Kim KH ;
Billadeau DD
作者单位:
Univ Illinois, Dept Med Chem & Pharmacognosy, Drug Discovery Program, Chicago, IL 60612 USA
[1]
Mayo Clin, Coll Med, Div Oncol Res, Rochester, MN 55905 USA
[2]
期刊:
《Journal of Medicinal Chemistry》
2008年51卷15期4370-4373页
关键词:
ISOFORM SELECTIVITY;PANCREATIC-CANCER;PROSTATE-CANCER;ACETYLATION;CELLS;NEUROPROTECTION;TRANSCRIPTION;COMBINATION;PROTEIN
发布时间:
2013-11-21
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