摘要在体皮肤药代动力学研究可以直接反应出药物在皮内的变化规律,是研究外用药及系统用药后,药物在靶部位作用强度、量-效关系、代谢规律的直接手段,有助于制定合理的给药剂量及间隔,为合理用药提供依据.实验的模型和方法主要包括胶带黏贴试验、皮肤微透析、吸疱试验、组织活检、琼脂凝胶板试验及光谱分析法等.
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abstractsIn vivo dermopharmacokinetic research can directly disclose the action intensity, dose-effect relationship, and metabolic rhythm of topical and systemic drugs in target sites, which will contribute to the scheduling of reasonable dosage and dosing interval and provide a basis for rational application of drugs. The methods for in vivo dermopharmacokinetic research include tape stripping, dermal microdialysis, suction blistering, biopsy, agar gel disc test, spectroscopic analysis, etc.
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