Discovery of Highly Selective Inhibitors of Calmodulin-Dependent Kinases That Restore Insulin Sensitivity in the Diet-Induced Obesity in Vivo Mouse Model
作者:
Fromont, Christophe [1]
;
Atzori, Alessio [2]
;
Kaur, Divneet [3]
;
Hashmi, Lubna [4]
;
Greco, Graziella [5]
;
Cabanillas, Alejandro [6]
;
Van Nguyen, Huy [7]
;
Jones, D. Heulyn [8]
;
Garzon, Miguel [9]
;
Varela, Ana [10]
;
Stevenson, Brett [11]
;
Iacobini, Greg P. [12]
;
Lenoir, Marc [13]
;
Rajesh, Sundaresan [14]
;
Box, Clare ;
Kumar, Jitendra ;
Grant, Paige ;
Novitskaya, Vera ;
Morgan, Juliet ;
Sorrell, Fiona J. ;
Redondo, Clara ;
Kramer, Andreas ;
Harris, C. John ;
Leighton, Brendan ;
Vickers, Steven P. ;
Cheetham, Sharon C. ;
Kenyon, Colin ;
Grabowska, Anna M. ;
Overduin, Michael ;
Berditchevski, Fedor ;
Weston, Chris J. ;
Knapp, Stefan ;
Fischer, Peter M. ;
Butterworth, Sam
作者单位:
Univ Birmingham, Inst Canc & Genom Sci, Birmingham B15 2TT, W Midlands, England
[1]
Res Network, Sandwich CT13 9NJ, Kent, England
[2]
Univ Oxford, Struct Genom Consortium, Oxford OX3 7DQ, England
[3]
CJH Consultants, Brockenhurst SO42 7UQ, Hants, England
[4]
Univ Birmingham, Coll Med & Dent Sci, Sch Pharm, Edgbaston B15 2TT, England
[5]
RenaSci Ltd, Nottingham NG1 1GF, England
[6]
Univ Manchester, Div Pharm & Optometry, Sch Hlth Sci, Manchester Acad Hlth Sci Ctr, Manchester M13 9PL, Lancs, England
[7]
Univ Nottingham, Ex Vivo Canc Pharmacol Ctr Excellence, Canc Biol, Div Canc & Stem Cells,Sch Med, Nottingham NG7 2RD, England
[8]
Univ Alberta, Dept Biochem, Edmonton, AB T6G 2H7, Canada
[9]
Univ Stellenbosch, DST NRF Ctr Excellence Biomed TB Res, SAMRC Ctr Mol & Cellular Biol, Div Mol Biol & Human Genet,Fac Med & Hlth Sci, ZA-8000 Cape Town, South Africa
[10]
Univ Nottingham, Ctr Biomol Sci, Nottingham NG7 2RD, England
[11]
Sygnature Discovery, Nottingham NG1 1GF, England
[12]
Univ Birmingham, Liver Res Ctr, Inst Immunol & Immunotherapy, Birmingham B15 2TT, W Midlands, England
[13]
Goethe Univ Frankfurt, Struct Genom Consortium, D-60438 Frankfurt, Germany
[14]
发布时间
2021-09-25
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Journal of Medicinal Chemistry
Journal of Medicinal Chemistry
6784-6801页
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