In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists

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作者： Romeo, Isabella ^[1] ; Brizzi, Antonella ^[2] ; Pessina, Federica ^[3] ; Ambrosio, Francesca Alessandra ^[4] ; Aiello, Francesca ^[5] ; Belardo, Carmela ^[6] ; Carullo, Gabriele ; Costa, Giosue ; De Petrocellis, Luciano ; Frosini, Maria ; Luongo, Livio ; Maramai, Samuele ; Paolino, Marco ; Moriello, Aniello Schiano ; Mugnaini, Claudia ; Scorzelli, Francesco ; Maione, Sabatino ; Corelli, Federico ; Di Marzo, Vincenzo ; Alcaro, Stefano ; Artese, Anna

作者单位： Univ Siena ^[1] Magna Graecia Univ Catanzaro ^[2] Univ Calabria ^[3] Univ Campania L Vanvitelli ^[4] CNR ^[5] Recipharm Edmond Pharm ^[6]

关键词 STRUCTURE-AFFINITY RELATIONSHIPS CAPSAICIN RECEPTOR TRPV1 VANILLOID TYPE-1 TRPV1 PHARMACOLOGICAL CHARACTERIZATION ION-CHANNEL LIGAND RESINIFERATOXIN BINDING IDENTIFICATION ACTIVATION

发布时间 2023-08-30

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准确一般字义偏差语意偏离译文作用小提交