A systematic strategy for estimating hERG block potency and its implications in a new cardiac safety paradigm (vol 394C, 114961, 2020)
作者:
Ridder, Bradley J. [1]
;
Leishman, Derek J. [2]
;
Bridgland-Taylor, Matthew [3]
;
Samieegohar, Mohammadreza [4]
;
Han, Xiaomei [5]
;
Wu, Wendy W. [6]
;
Randolph, Aaron [7]
;
Tran, Phu [8]
;
Sheng, Jiansong [9]
;
Danker, Timm [10]
;
Lindqvist, Anders [11]
;
Konrad, Daniel [12]
;
Hebeisen, Simon [13]
;
Polonchuk, Liudmila [14]
;
Gissinger, Evgenia [15]
;
Renganathan, Muthukrishnan [16]
;
Koci, Bryan [17]
;
Wei, Haiyang [18]
;
Fan, Jingsong ;
Levesque, Paul ;
Kwagh, Jae ;
Imredy, John ;
Zhai, Jin ;
Rogers, Marc ;
Humphries, Edward ;
Kirby, Robert ;
Stoelzle-Feix, Sonja ;
Brinkwirth, Nina ;
Rotordam, Maria Giustina ;
Becker, Nadine ;
Friis, Soren ;
Rapedius, Markus ;
Goetze, Tom A. ;
Strassmaier, Tim ;
Okeyo, George ;
Kramer, James ;
Kuryshev, Yuri ;
Wu, Caiyun ;
Himmel, Herbert ;
Mirams, Gary R. ;
Strauss, David G. ;
Bardenet, Remi ;
Li, Zhihua
作者单位:
Eurofins Discovery, Eurofins Sci, 6 Res Pk Dr, St Charles, MO 63304 USA
[1]
F Hoffmann La Roche Ltd, F Hoffmann La Roche AG, Bldg 73 R 103b Grenzacherstr,124, CH-4070 Basel
[2]
NMI TT GmbH, Markwiesenstr 55, D-72770 Reutlingen, Germany
[3]
Nan Technol USA, 1 Naylon Pl,Suite C, Livingston, NJ 07039 USA
[4]
AstraZeneca, Clin Pharmacol & Safety Sci, Biopharmaceut R&D, Cambridge, England
[5]
Univ Lille, CNRS, Cent Lille, UMR 9189,CRIStAL, Villeneuve Dascq, France
[6]
Bayer AG, RD TS TOX SP SPL1,Aprather Weg 18a, D-42096 Wuppertal, Germany
[7]
Eli Lilly & Co, Dept Toxicol & Pathol, Indianapolis, IN 46285 USA
[8]
Ion Channel Co, BSYS GmbH, Benkenstr 254, CH-4108 Witterswil, Switzerland
[9]
CiPA LAB, 900 Clopper Rd,Suite 130, Gaithersburg, MD 20878 USA
[10]
Charles River Labs, 14656 Neo Pkwy, Cleveland, OH 44128 USA
[11]
Metr Biosci Ltd, Riverside 3,Suite 1,Granta Pk, Cambridge CB21 6AD, England
[12]
US FDA, Div Appl Regulatory Sci, Off Clin Pharmacol, Off Translat Sci,Ctr Drug Evaluat & Res, 10903
[13]
Soph Biosc AS, Baltorpvej 154, DK-2750 Ballerup, Denmark
[14]
Merck & Co Inc, Kenilworth, NJ USA
[15]
Bristol Myers Squibb, Bristol Myers Squibb Co, Discovery Toxicol, 3551 Lawrenceville,Princeton Rd
[16]
Univ Nottingham, Ctr Math Med & Biol, Sch Math Sci, Nottingham, England
[17]
Nan Technol Munich, Ganghoferstr 70A, D-80339 Munich, Germany
[18]
发布时间
2021-07-24
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