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The promise and peril of chemical probes

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作者单位: Univ Oxford, Struct Genom Consortium, Oxford, England [1] Simon Fraser Univ, Dept Chem, Burnaby, BC V5A 1S6, Canada [2] Pfizer, Worldwide Med Chem, Cambridge, MA USA [3] Struct Genom Consortium, Toronto, ON, Canada [4] Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England [5] Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA [6] Epizyme Inc, Cambridge, MA USA [7] Janssen Res & Dev, Spring House, PA USA [8] Karolinska Inst, Struct Genom Consortium, Solna, Sweden [9] Univ N Carolina, Eshelman Sch Pharm, Chapel Hill, NC USA [10] Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA [11] Austrian Acad Sci, CeMM Res Ctr Mol Med, A-1010 Vienna, Austria [12] Univ Calif San Francisco, Sch Pharm, San Francisco, CA 94143 USA [13] Constellat Pharmaceut, Cambridge, MA USA [14] Broad Inst, Ctr Sci Therapeut, Cambridge, MA USA [15] Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON, Canada [16] NIH, Natl Ctr Adv Translat Sci, Bethesda, MD 20892 USA [17] Mayo Clin, Coll Med, Dept Mol Pharmacol & Expt Therapeut, Rochester, MN USA [18] Takeda Calif Inc, San Diego, CA USA [19] Univ Minnesota, Minneapolis, MN USA [20] GlaxoSmithKline, Collegeville, PA USA [21] Harvard Univ, Dept Biol Chem & Mol Pharmacol, Cambridge, MA 02138 USA [22] Scripps Res Inst, Dept Physiol Chem, San Diego, CA USA [23] Merck Res Labs, Oncol Discovery, Boston, MA USA [24] Bayer Pharma AG, Berlin, Germany [25] Janssen Res & Dev, High Wycombe, Bucks, England [26] Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94143 USA [27] Monash Univ, Fac Pharm & Pharmaceut Sci, Melbourne, Vic 3004, Australia [28] Merck Res Labs, Discovery Chem, Boston, MA USA [29] Univ N Carolina, Eshelman Sch Pharm, Ctr Integrat Chem Biol & Drug Discovery, Div Chem Biol & Med Chem, Chapel Hill, NC USA [30] Vertex Pharmaceut, Boston, MA USA [31] European Bioinformat Inst, European Mol Biol Lab, Hinxton, England [32] AbbVie, N Chicago, IL USA [33] Boehringer Ingelheim GmbH & Co KG, Corp Dept Res Networking, Ingelheim, Germany [34] Univ Dundee, Sir James Black Ctr, Dundee, Scotland [35] GlaxoSmithKline, Canc Epigenet, Collegeville, PA USA [36] McGill Univ, Struct Genom Consortium, Montreal, PQ, Canada [37] CHDI Fdn, CHDI Management, Los Angeles, CA USA [38]
发布时间 2015-09-29
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Nature chemical biology

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