The staurosporine-like compound L-753,000 (NB-506) potentiates the neurotrophic effects of neurotrophin-3 by acting selectively at the TrkA receptor.
第一作者:
S,Pollack
第一单位:
Department of Biochemistry, Merck Sharp and Dohme Research Laboratories, Neuroscience Research Centre, Harlow, Essex, United Kingdom. scott_pollack@merck.com
作者:
医学主题词
方差分析(Analysis of Variance);动物(Animals);CHO细胞(CHO Cells);钙-钙调素依赖性蛋白激酶类(Calcium-Calmodulin-Dependent Protein Kinases);卡唑类(Carbazoles);细胞, 培养的(Cells, Cultured);鸡胚(Chick Embryo);鸡(Chickens);仓鼠亚科(Cricetinae);药物协同作用(Drug Synergism);酶激活(Enzyme Activation);酶抑制剂(Enzyme Inhibitors);葡糖苷类(Glucosides);吲哚生物碱类(Indole Alkaloids);神经生长因子类(Nerve Growth Factors);神经突(Neurites);神经元(Neurons);神经营养因子3(Neurotrophin 3);蛋白激酶C(Protein Kinase C);原癌基因蛋白质类(Proto-Oncogene Proteins);大鼠(Rats);受体蛋白质酪氨酸激酶类(Receptor Protein-Tyrosine Kinases);受体, trkA(Receptor, trkA);受体, 神经生长因子类(Receptors, Nerve Growth Factor);星状孢子素(Staurosporine)
DOI
10.1124/mol.56.1.185
PMID
10385700
发布时间
2019-06-07
- 浏览19
Molecular pharmacology
185-95页
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