Design and synthesis of novel alpha(1)(a) adrenoceptor-selective antagonists. 1. Structure-activity relationship in dihydropyrimidinones.
作者:
主题词
肾上腺素能α-1受体拮抗剂(Adrenergic alpha-1 Receptor Antagonists);肾上腺素能α拮抗剂(Adrenergic alpha-Antagonists);动物(Animals);结合, 竞争性(Binding, Competitive);血压(Blood Pressure);狗(Dogs);药物设计(Drug Design);药物评价, 临床前(Drug Evaluation, Preclinical);人类(Humans);男(雄)性(Male);前列腺(Prostate);嘧啶酮类(Pyrimidinones);放射配体测定(Radioligand Assay);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 肾上腺素能α1(Receptors, Adrenergic, alpha-1);立体异构现象(Stereoisomerism);尿道(Urethra)
DOI
10.1021/jm990200p
PMID
10579840
发布时间
2019-07-09
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