Residue Gly1326 of the N-type calcium channel alpha 1B subunit controls reversibility of omega-conotoxin GVIA and MVIIA block.
第一作者:
Z P,Feng
第一单位:
Departments of Physiology & Biophysics and Pharmacology & Therapeutics, Neuroscience Research Group, University of Calgary, Calgary, Alberta T2N 4N1, Canada.
作者:
医学主题词
氨基酸序列(Amino Acid Sequence);氨基酸取代(Amino Acid Substitution);精氨酸(Arginine);结合部位(Binding Sites);钙(Calcium);钙通道阻滞药(Calcium Channel Blockers);钙通道, N型(Calcium Channels, N-Type);细胞系(Cell Line);谷氨酸(Glutamic Acid);甘氨酸(Glycine);人类(Humans);动力学(Kinetics);膜电位(Membrane Potentials);模型, 分子(Models, Molecular);分子序列数据(Molecular Sequence Data);诱变, 定点(Mutagenesis, Site-Directed);膜片钳术(Patch-Clamp Techniques);脯氨酸(Proline);蛋白质结构, 二级(Protein Structure, Secondary);蛋白质亚单位(Protein Subunits);转染(Transfection);ω蜗牛毒素GVIA(omega-Conotoxin GVIA);ω蜗牛毒素类(omega-Conotoxins)
DOI
10.1074/jbc.M100406200
PMID
11279062
发布时间
2021-02-09
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