UCN-01 (7-hydoxystaurosporine) inhibits in vivo growth of human cancer cells through selective perturbation of G1 phase checkpoint machinery.
第一作者:
S,Abe
第一单位:
Department of Surgery, School of Medicine, Keio University, Shinjuku-ku, Tokyo 160-8582, Japan.
作者:
医学主题词
生物碱类(Alkaloids);动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);印迹法, 蛋白质(Blotting, Western);乳腺肿瘤(Breast Neoplasms);CDC2-CDC28激酶类(CDC2-CDC28 Kinases);细胞分裂(Cell Division);细胞周期蛋白依赖激酶2(Cyclin-Dependent Kinase 2);周期素依赖激酶抑制剂p21(Cyclin-Dependent Kinase Inhibitor p21);细胞周期蛋白质依赖激酶类(Cyclin-Dependent Kinases);细胞周期蛋白类(Cyclins);DNA, 肿瘤(DNA, Neoplasm);抗药性, 肿瘤(Drug Resistance, Neoplasm);G1期(G1 Phase);人类(Humans);免疫组织化学(Immunohistochemistry);男(雄)性(Male);小鼠(Mice);小鼠, 近交BALB C(Mice, Inbred BALB C);小鼠, 裸(Mice, Nude);肿瘤移植(Neoplasm Transplantation);肿瘤, 实验性(Neoplasms, Experimental);胰腺肿瘤(Pancreatic Neoplasms);磷酰化(Phosphorylation);视网膜母细胞瘤蛋白质(Retinoblastoma Protein);星状孢子素(Staurosporine);移植, 异种(Transplantation, Heterologous)
DOI
10.1111/j.1349-7006.2001.tb01127.x
PMID
11376563
发布时间
2021-12-03
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