Computer-assisted mutagenesis of ecotin to engineer its secondary binding site for urokinase inhibition.
第一作者:
Martha C A,Laboissière
第一单位:
Departamento de Ciências Farmacêuticas, Faculdade de Ciências da Saúde, Universidade de Brasilia, Campus Universitário Darcy Ribeiro, 70910-900 Brasilia, DF Brasil.
作者:
医学主题词
氨基酸取代(Amino Acid Substitution);细菌蛋白质类(Bacterial Proteins);结合部位(Binding Sites);大肠杆菌(Escherichia coli);大肠杆菌蛋白质类(Escherichia coli Proteins);遗传工程(Genetic Engineering);动力学(Kinetics);模型, 分子(Models, Molecular);诱变(Mutagenesis);肽库(Peptide Library);胞质蛋白质类(Periplasmic Proteins);蛋白质结合(Protein Binding);尿激酶型纤溶酶原激活物(Urokinase-Type Plasminogen Activator)
DOI
10.1074/jbc.M203076200
PMID
11959867
发布时间
2021-02-06
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