[99mTc]Demotate, a new 99mTc-based [Tyr3]octreotate analogue for the detection of somatostatin receptor-positive tumours: synthesis and preclinical results.
第一作者:
Theodosia,Maina
第一单位:
Institute of Radioisotopes - Radiodiagnostic Products, National Center for Scientific Research Demokritos, 15310 Ag. Paraskevi, Attikis, Athens, Greece. mainathe@mail.demokritos.gr
作者:
主题词
动物(Animals);大脑皮质(Cerebral Cortex);女(雌)性(Female);同位素标记(Isotope Labeling);男(雄)性(Male);代谢清除率(Metabolic Clearance Rate);小鼠(Mice);小鼠, 裸(Mice, Nude);模型, 化学(Models, Chemical);奥曲肽(Octreotide);有机锝化合物(Organotechnetium Compounds);胰腺肿瘤(Pancreatic Neoplasms);肽类, 环(Peptides, Cyclic);蛋白质结合(Protein Binding);放射性核素显像(Radionuclide Imaging);大鼠(Rats);大鼠, Wistar(Rats, Wistar);受体, 生长抑素(Receptors, Somatostatin);结果可重复性(Reproducibility of Results);敏感性与特异性(Sensitivity and Specificity);组织分布(Tissue Distribution);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1007/s00259-002-0782-9
PMID
12029547
发布时间
2018-09-24
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