Effect of albumin and cytosol on enzyme kinetics of tolbutamide hydroxylation and on inhibition of CYP2C9 by gemfibrozil in human liver microsomes.
第一作者:
Jun-Sheng,Wang
第一单位:
Department of Clinical Pharmacology, University of Helsinki and Helsinki University Central Hospital, Haartmaninkatu 4, FIN-00290 Helsinki, Finland.
作者:
医学主题词
白蛋白类(Albumins);算法(Algorithms);芳基烃羟化酶类(Aryl Hydrocarbon Hydroxylases);色谱法, 高压液相(Chromatography, High Pressure Liquid);胞质溶胶(Cytosol);酶抑制剂(Enzyme Inhibitors);吉非贝齐(Gemfibrozil);人类(Humans);羟基化(Hydroxylation);降血糖药(Hypoglycemic Agents);降血脂药物(Hypolipidemic Agents);动力学(Kinetics);微粒体, 肝(Microsomes, Liver);类固醇16-α-羟化酶(Steroid 16-alpha-Hydroxylase);甾类羟化酶类(Steroid Hydroxylases);甲苯磺丁脲(Tolbutamide)
DOI
10.1124/jpet.302.1.43
PMID
12065698
发布时间
2025-03-06
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