Novel dual inhibitors of AChE and MAO derived from hydroxy aminoindan and phenethylamine as potential treatment for Alzheimer's disease.
作者:
主题词
乙酰胆碱酯酶(Acetylcholinesterase);阿尔茨海默病(Alzheimer Disease);动物(Animals);结合部位(Binding Sites);丁酰胆碱酯酶(Butyrylcholinesterase);氨甲酸酯类(Carbamates);牛(Cattle);胆碱酯酶抑制剂(Cholinesterase Inhibitors);人类(Humans);茚满类(Indans);模型, 分子(Models, Molecular);单胺氧化酶(Monoamine Oxidase);单胺氧化酶抑制剂(Monoamine Oxidase Inhibitors);帕吉林(Pargyline);苯乙胺类(Phenethylamines);丙胺类(Propylamines);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm020120c
PMID
12431053
发布时间
2019-07-10
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