Design and synthesis of 8-hydroxy-[1,6]naphthyridines as novel inhibitors of HIV-1 integrase in vitro and in infected cells.
作者:
主题词
投药, 口服(Administration, Oral);动物(Animals);抗HIV药(Anti-HIV Agents);细胞系(Cell Line);HIV整合酶抑制剂(HIV Integrase Inhibitors);HIV-1(HIV-1);人类(Humans);注射, 静脉内(Injections, Intravenous);萘啶类(Naphthyridines);大鼠(Rats);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm025553u
PMID
12570367
发布时间
2004-11-17
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