MCC-134, a single pharmacophore, opens surface ATP-sensitive potassium channels, blocks mitochondrial ATP-sensitive potassium channels, and suppresses preconditioning.
作者:
主题词
腺苷三磷酸(Adenosine Triphosphate);动物(Animals);强心药(Cardiotonic Agents);细胞膜(Cell Membrane);细胞, 培养的(Cells, Cultured);二氮嗪(Diazoxide);导电性(Electric Conductivity);女(雌)性(Female);黄素蛋白类(Flavoproteins);荧光(Fluorescence);心脏(Heart);咪唑类(Imidazoles);缺血预处理, 心肌(Ischemic Preconditioning, Myocardial);男(雄)性(Male);小鼠(Mice);线粒体, 心脏(Mitochondria, Heart);心肌梗死(Myocardial Infarction);膜片钳术(Patch-Clamp Techniques);钾通道阻滞剂(Potassium Channel Blockers);钾通道(Potassium Channels);兔(Rabbits);硫代酰胺类(Thioamides)
DOI
10.1161/01.cir.0000051457.64240.63
PMID
12615799
发布时间
2019-06-23
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Circulation
1183-8页
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