Small molecule LFA-1 antagonists compete with an anti-LFA-1 monoclonal antibody for binding to the CD11a I domain: development of a flow-cytometry-based receptor occupancy assay.
第一作者:
Joseph R,Woska
第一单位:
Department of Biology, Boehringer Ingelheim Pharmaceuticals, Inc., 900 Ridgebury Rd., P.O. Box 368, Ridgefield, CT 06877, USA. jwoska@rdg.boehringer-ingelheim.com
作者:
主题词
动物(Animals);抗体, 单克隆(Antibodies, Monoclonal);抗体特异性(Antibody Specificity);结合, 竞争性(Binding, Competitive);细胞黏附分子(Cell Adhesion Molecules);流式细胞术(Flow Cytometry);人类(Humans);咪唑类(Imidazoles);咪唑啉啶类(Imidazolidines);淋巴细胞功能相关抗原1(Lymphocyte Function-Associated Antigen-1);淋巴细胞(Lymphocytes);中性白细胞(Neutrophils);黑猩猩属(Pan troglodytes);受体, 白细胞黏附(Receptors, Leukocyte-Adhesion);松鼠猴属(Saimiri)
DOI
10.1016/s0022-1759(03)00176-5
PMID
12799043
发布时间
2019-12-10
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