Design, synthesis, and biological evaluation of cytotoxic 11-alkenylindenoisoquinoline topoisomerase I inhibitors and indenoisoquinoline-camptothecin hybrids.
作者:
主题词
抗肿瘤药(Antineoplastic Agents);喜树碱(Camptothecin);DNA拓扑异构酶类, Ⅰ型(DNA Topoisomerases, Type I);药物设计(Drug Design);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);异喹啉类(Isoquinolines);磁共振波谱学(Magnetic Resonance Spectroscopy);模型, 分子(Models, Molecular);构效关系(Structure-Activity Relationship);拓扑异构酶I抑制剂(Topoisomerase I Inhibitors);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1021/jm0300476
PMID
12852757
发布时间
2013-11-21
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