A high-throughput, nonisotopic, competitive binding assay for kinases using nonselective inhibitor probes (ED-NSIP).
作者:
主题词
腺苷三磷酸(Adenosine Triphosphate);动物(Animals);结合部位(Binding Sites);结合, 竞争性(Binding, Competitive);组合化学技术(Combinatorial Chemistry Techniques);二甲亚砜(Dimethyl Sulfoxide);药物评价, 临床前(Drug Evaluation, Preclinical);酶抑制剂(Enzyme Inhibitors);糖原合成酶激酶3(Glycogen Synthase Kinase 3);人类(Humans);同位素(Isotopes);分子生物学(Molecular Biology);蛋白激酶抑制剂(Protein Kinase Inhibitors);蛋白激酶类(Protein Kinases);重组蛋白质类(Recombinant Proteins);结果可重复性(Reproducibility of Results);星状孢子素(Staurosporine);β半乳糖苷酶类(beta-Galactosidase)
DOI
10.1177/1087057102238624
PMID
14599348
发布时间
2021-12-03
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