Orally active anti-proliferation agents: novel diphenylamine derivatives as FGF-R2 autophosphorylation inhibitors.
第一作者:
Toshiyuki,Shimizu
第一单位:
Pharmaceutical Research Laboratories, Kirin Brewery Co., Ltd., 3 Miyahara, Takasaki, Gunma, 370-1295, Japan. tshimuzu@kirin.co.jp
作者:
主题词
投药, 口服(Administration, Oral);动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞分裂(Cell Division);细胞系, 肿瘤(Cell Line, Tumor);二苯胺(Diphenylamine);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);分子结构(Molecular Structure);磷酰化(Phosphorylation);大鼠(Rats);受体蛋白质酪氨酸激酶类(Receptor Protein-Tyrosine Kinases);受体, 成纤维细胞生长因子, 2型(Receptor, Fibroblast Growth Factor, Type 2);受体, 成纤维细胞生长因子(Receptors, Fibroblast Growth Factor);胃肿瘤(Stomach Neoplasms)
DOI
10.1016/j.bmcl.2003.12.019
PMID
15012985
发布时间
2013-11-21
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