The cyclooxygenase-2 inhibitor GW406381X [2-(4-ethoxyphenyl)-3-[4-(methylsulfonyl)phenyl]-pyrazolo[1,5-b]pyridazine] is effective in animal models of neuropathic pain and central sensitization.
作者:
主题词
动物(Animals);脑(Brain);COS细胞(COS Cells);辣椒辣素(Capsaicin);环加氧酶抑制药(Cyclooxygenase Inhibitors);疾病模型, 动物(Disease Models, Animal);剂量效应关系, 药物(Dose-Response Relationship, Drug);人类(Humans);烃类, 芳香(Hydrocarbons, Aromatic);痛觉过敏(Hyperalgesia);男(雄)性(Male);小鼠(Mice);氮(Nitrogen);疼痛(Pain);吡唑类(Pyrazoles);哒嗪类(Pyridazines);大鼠(Rats)
DOI
10.1124/jpet.104.075267
PMID
15572651
发布时间
2022-03-09
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