Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles.
第一作者:
J P,Mallamo
第一单位:
Department of Medicinal Chemistry, Sterling Winthrop Pharmaceuticals Research Division, Rensselaer, New York 12144.
作者:
医学主题词
雄激素拮抗药(Androgen Antagonists);雄激素受体拮抗剂(Androgen Receptor Antagonists);电化学(Electrochemistry);杂环化合物(Heterocyclic Compounds);受体, 雄激素(Receptors, Androgen);底物特异性(Substrate Specificity);X线衍射(X-Ray Diffraction)
DOI
10.1021/jm00088a001
PMID
1588549
发布时间
2019-07-09
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