Use of structure-based drug design approaches to obtain novel anthranilic acid acyl carrier protein synthase inhibitors.
作者:
主题词
抗菌药(Anti-Bacterial Agents);色谱法, 高压液相(Chromatography, High Pressure Liquid);结晶学, X线(Crystallography, X-Ray);药物设计(Drug Design);抗药性, 细菌(Drug Resistance, Bacterial);革兰氏阳性菌(Gram-Positive Bacteria);配体(Ligands);微生物敏感性试验(Microbial Sensitivity Tests);模型, 分子(Models, Molecular);分子结构(Molecular Structure);量化构效关系(Quantitative Structure-Activity Relationship);立体异构现象(Stereoisomerism);转移酶类(其他取代磷酸族)(Transferases (Other Substituted Phosphate Groups))
DOI
10.1021/jm050523n
PMID
16335920
发布时间
2012-11-15
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