Polymer-supported synthesis of pyridone-focused libraries as inhibitors of anaplastic lymphoma kinase.
第一作者:
Tong,Zhu
第一单位:
Department of High Throughput Medicinal Chemistry, ChemBridge Research Laboratories, San Diego, California 92127, USA.
作者:
医学主题词
组合化学技术(Combinatorial Chemistry Techniques);药物设计(Drug Design);酶抑制剂(Enzyme Inhibitors);模型, 化学(Models, Chemical);聚合物(Polymers);蛋白酪氨酸激酶类(Protein-Tyrosine Kinases);吡啶酮类(Pyridones);受体蛋白质酪氨酸激酶类(Receptor Protein-Tyrosine Kinases);立体异构现象(Stereoisomerism);工艺学, 制药(Technology, Pharmaceutical)
DOI
10.1021/cc060018r
PMID
16677010
发布时间
2018-12-01
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