Synthesis and pharmacological characterization of nicotinic acetylcholine receptor properties of (+)- and (-)-pyrido-[3,4-b]homotropanes.
作者:
主题词
镇痛药(Analgesics);动物(Animals);细胞系(Cell Line);大脑皮质(Cerebral Cortex);结晶学, X线(Crystallography, X-Ray);辨别学习(Discrimination Learning);男(雄)性(Male);神经元(Neurons);尼古丁(Nicotine);烟碱激动剂(Nicotinic Agonists);烟碱拮抗剂(Nicotinic Antagonists);疼痛测定(Pain Measurement);膜片钳术(Patch-Clamp Techniques);吡啶类(Pyridines);放射配体测定(Radioligand Assay);大鼠(Rats);受体, 烟碱(Receptors, Nicotinic);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship);托烷类(Tropanes)
DOI
10.1021/jm060122n
PMID
16722642
发布时间
2015-11-19
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