A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening.
作者:
主题词
氨肽酶类(Aminopeptidases);动物(Animals);组合化学技术(Combinatorial Chemistry Techniques);药物设计(Drug Design);药物评价, 临床前(Drug Evaluation, Preclinical);酶激活(Enzyme Activation);羟肟酸类(Hydroxamic Acids);肾(Kidney);微粒体(Microsomes);分子结构(Molecular Structure);蛋白酶抑制药(Protease Inhibitors);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship);猪(Swine);锌(Zinc)
DOI
10.1016/j.bmc.2006.10.010
PMID
17070058
发布时间
2013-11-21
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