Synthesis and structure-activity relationships of spirohydantoin-derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1).
作者:
主题词
减肥药(Anti-Obesity Agents);药物设计(Drug Design);人类(Humans);乙内酰脲类(Hydantoins);动力学(Kinetics);蛋白质结合(Protein Binding);受体, 垂体激素(Receptors, Pituitary Hormone);螺环化合物(Spiro Compounds);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2007.01.104
PMID
17350839
发布时间
2007-12-03
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