Potent nonpeptide antagonists of the bradykinin B1 receptor: structure-activity relationship studies with novel diaminochroman carboxamides.
作者:
主题词
酰胺类(Amides);镇痛药(Analgesics);动物(Animals);苯吡喃类(Benzopyrans);血压(Blood Pressure);CHO细胞(CHO Cells);钙(Calcium);色满类(Chromans);仓鼠亚科(Cricetinae);仓鼠属(Cricetulus);人类(Humans);炎症(Inflammation);男(雄)性(Male);微粒体(Microsomes);疼痛(Pain);兔(Rabbits);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 缓激肽B1(Receptor, Bradykinin B1);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship);磺胺类(Sulfonamides)
DOI
10.1021/jm070055c
PMID
17408249
发布时间
2014-11-20
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Journal of medicinal chemistry
2200-12页
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