Synthesis, structure-activity relationship and in vivo antiinflammatory efficacy of substituted dipiperidines as CCR2 antagonists.
作者:
主题词
动物(Animals);消炎药, 非甾类(Anti-Inflammatory Agents, Non-Steroidal);关节炎, 实验性(Arthritis, Experimental);哮喘(Asthma);细胞系(Cell Line);趋化作用(Chemotaxis);结晶学, X线(Crystallography, X-Ray);人类(Humans);男(雄)性(Male);小鼠(Mice);哌啶类(Piperidines);大鼠(Rats);大鼠, 近交Lew(Rats, Inbred Lew);受体, CCR2(Receptors, CCR2);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm070902b
PMID
17929797
发布时间
2007-11-08
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