Phenylpiperidine-benzoxazinones as urotensin-II receptor antagonists: synthesis, SAR, and in vivo assessment.
第一作者:
Diane K,Luci
第一单位:
Research & Early Development, Johnson & Johnson Pharmaceutical Research & Development, Welsh and McKean Roads, Spring House, PA 19477-0776, USA.
作者:
主题词
动物(Animals);苯并恶嗪类(Benzoxazines);CHO细胞(CHO Cells);仓鼠亚科(Cricetinae);仓鼠属(Cricetulus);人类(Humans);哌啶类(Piperidines);大鼠(Rats);受体, G-蛋白偶联(Receptors, G-Protein-Coupled);构效关系(Structure-Activity Relationship);尿紧张素类(Urotensins)
DOI
10.1016/j.bmcl.2007.09.092
PMID
17933531
发布时间
2007-11-06
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