Effect of bradykinin metabolism inhibitors on evoked hypotension in rats: rank efficacy of enzymes associated with bradykinin-mediated angioedema.
第一作者:
R M,Fryer
第一单位:
Department of Integrative Pharmacology, Global Pharmaceutical Research and Development, Abbott Laboratories, Abbott Park, IL 60064-6119, USA. ryan.fryer@abbott.com
作者:
医学主题词
氨肽酶类(Aminopeptidases);血管性水肿(Angioedema);血管紧张素转换酶抑制药(Angiotensin-Converting Enzyme Inhibitors);动物(Animals);缓激肽(Bradykinin);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物评价, 临床前(Drug Evaluation, Preclinical);酶抑制剂(Enzyme Inhibitors);低血压(Hypotension);茚满类(Indans);赖诺普利(Lisinopril);男(雄)性(Male);脑啡肽酶(Neprilysin);肽类(Peptides);丙酸盐类(Propionates);吡啶类(Pyridines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);硫氮杂|艹卓|类(Thiazepines)
DOI
10.1038/sj.bjp.0707641
PMID
18084312
发布时间
2022-03-11
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