Exploration of the internal cavity of histone deacetylase (HDAC) with selective HDAC1/HDAC2 inhibitors (SHI-1:2).
作者:
主题词
苯衍生物(Benzene Derivatives);结合部位(Binding Sites);组蛋白脱乙酰基酶1(Histone Deacetylase 1);组蛋白脱乙酰基酶2(Histone Deacetylase 2);组蛋白脱乙酰基酶抑制剂(Histone Deacetylase Inhibitors);组蛋白脱乙酰基酶类(Histone Deacetylases);人类(Humans);模型, 分子(Models, Molecular);分子结构(Molecular Structure);蛋白质亚型(Protein Isoforms);阻遏蛋白质类(Repressor Proteins);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2007.12.031
PMID
18182289
发布时间
2009-11-19
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