Synthesis and biological evaluation of 99mTc, Re-monoamine-monoamide conjugated to 2-(4-aminophenyl)benzothiazole as potential probes for beta-amyloid plaques in the brain.
第一作者:
Xiangji,Chen
第一单位:
Key Laboratory of Radiopharmaceuticals, (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University, Beijing 100875, PR China.
作者:
主题词
阿尔茨海默病(Alzheimer Disease);酰胺类(Amides);胺类(Amines);淀粉样β肽类(Amyloid beta-Peptides);动物(Animals);苯并噻唑类(Benzothiazoles);血脑屏障(Blood-Brain Barrier);脑(Brain);人类(Humans);同位素标记(Isotope Labeling);男(雄)性(Male);小鼠(Mice);显微镜检查, 荧光(Microscopy, Fluorescence);中年人(Middle Aged);有机锝化合物(Organotechnetium Compounds);放射性核素显像(Radionuclide Imaging);放射性药物(Radiopharmaceuticals);铼(Rhenium);锝化合物(Technetium Compounds);组织分布(Tissue Distribution)
DOI
10.1016/j.bmcl.2007.12.071
PMID
18191400
发布时间
2016-11-24
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