Pharmacological evaluation of LH-21, a newly discovered molecule that binds to cannabinoid CB1 receptor.
作者:
主题词
动物(Animals);减肥药(Anti-Obesity Agents);结合, 竞争性(Binding, Competitive);血脑屏障(Blood-Brain Barrier);CHO细胞(CHO Cells);仓鼠亚科(Cricetinae);仓鼠属(Cricetulus);环AMP(Cyclic AMP);环己醇类(Cyclohexanols);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物反向激动作用(Drug Inverse Agonism);进食(Eating);人类(Humans);注射, 腹腔内(Injections, Intraperitoneal);注射, 静脉内(Injections, Intravenous);男(雄)性(Male);小鼠(Mice);小鼠, 近交C57BL(Mice, Inbred C57BL);小鼠, 基因敲除(Mice, Knockout);蛋白质结合(Protein Binding);放射配体测定(Radioligand Assay);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 大麻酚, CB1(Receptor, Cannabinoid, CB1);受体, 大麻酚, CB2(Receptor, Cannabinoid, CB2);重组蛋白质类(Recombinant Proteins);转染(Transfection);三唑类(Triazoles);体重增长(Weight Gain)
DOI
10.1016/j.ejphar.2008.02.029
PMID
18336811
发布时间
2013-11-21
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