Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads.
作者:
主题词
化学, 药物(Chemistry, Pharmaceutical);二肽酶类(Dipeptidases);二肽类(Dipeptides);二肽基肽酶类和三肽基肽酶类(Dipeptidyl-Peptidases and Tripeptidyl-Peptidases);药物设计(Drug Design);酶抑制剂(Enzyme Inhibitors);人类(Humans);半数抑制浓度(Inhibitory Concentration 50);赖氨酸(Lysine);模型, 化学(Models, Chemical);分子结构(Molecular Structure);腈类(Nitriles);肽类(Peptides);吡咯烷类(Pyrrolidines);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2008.05.080
PMID
18556199
发布时间
2013-11-21
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