Rational design and synthesis of 2,2-bisheterocycle tandem derivatives as non-nucleoside hepatitis B virus inhibitors.
第一作者:
Hai-Jun,Chen
第一单位:
Chinese National Center for Drug Screening, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, 189 Guo Shou Jing Road, Shanghai 201203, China. fjnan@mail.shcnc.ac.cn
作者:
医学主题词
抗病毒药(Antiviral Agents);药物设计(Drug Design);乙型肝炎病毒(Hepatitis B virus);微生物敏感性试验(Microbial Sensitivity Tests);分子结构(Molecular Structure);小分子化合物库(Small Molecule Libraries);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship);噻唑类(Thiazoles);病毒非结构蛋白质类(Viral Nonstructural Proteins);病毒复制(Virus Replication)
DOI
10.1002/cmdc.200800136
PMID
18663717
发布时间
2016-11-24
- 浏览4
ChemMedChem
1316-21页
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