Novel acetylcholine and carbamoylcholine analogues: development of a functionally selective alpha4beta2 nicotinic acetylcholine receptor agonist.
第一作者:
Camilla P,Hansen
第一单位:
Department of Medicinal Chemistry, Faculty of Pharmaceutical Sciences, University of Copenhagen, UniVersitetsparken 2, DK-2100 Copenhagen Ø, Denmark.
作者:
医学主题词
乙酰胆碱(Acetylcholine);结合部位(Binding Sites);卡巴胆碱(Carbachol);细胞系(Cell Line);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物评价, 临床前(Drug Evaluation, Preclinical);人类(Humans);配体(Ligands);分子结构(Molecular Structure);烟碱激动剂(Nicotinic Agonists);受体, 烟碱(Receptors, Nicotinic);重组蛋白质类(Recombinant Proteins);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm701625v
PMID
18989912
发布时间
2015-11-19
- 浏览18
相似文献
- 中文期刊
- 外文期刊
- 学位论文
- 会议论文


换一批



