Synthesis and structure-activity relationship of 7-azaindole piperidine derivatives as CCR2 antagonists.
作者:
主题词
醇类(Alcohols);结合部位(Binding Sites);化学, 药物(Chemistry, Pharmaceutical);趋化因子CCL2(Chemokine CCL2);药物设计(Drug Design);人类(Humans);吲哚类(Indoles);半数抑制浓度(Inhibitory Concentration 50);分子结构(Molecular Structure);哌啶类(Piperidines);受体, CCR2(Receptors, CCR2);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2008.10.061
PMID
18990568
发布时间
2012-11-15
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