Design, structure-activity relationships and in vivo characterization of 4-amino-3-benzimidazol-2-ylhydroquinolin-2-ones: a novel class of receptor tyrosine kinase inhibitors.
作者:
主题词
动物(Animals);色谱法, 高压液相(Chromatography, High Pressure Liquid);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物设计(Drug Design);人类(Humans);磁共振波谱学(Magnetic Resonance Spectroscopy);质谱分析法(Mass Spectrometry);小鼠(Mice);小鼠, 近交NOD(Mice, Inbred NOD);小鼠, SCID(Mice, SCID);模型, 分子(Models, Molecular);蛋白激酶抑制剂(Protein Kinase Inhibitors);喹诺酮类(Quinolones);受体蛋白质酪氨酸激酶类(Receptor Protein-Tyrosine Kinases);构效关系(Structure-Activity Relationship)
DOI
10.1021/jm800790t
PMID
19113866
发布时间
2009-11-19
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