In vitro and in vivo activity of novel small-molecule inhibitors targeting the pleckstrin homology domain of protein kinase B/AKT.
第一作者:
Sylvestor A,Moses
第一单位:
Department of Molecular and Cellular Biology, The University of Arizona, Tucson, Arizona 85721-0038, USA.
作者:
医学主题词
动物(Animals);血蛋白质类(Blood Proteins);细胞系, 肿瘤(Cell Line, Tumor);女(雌)性(Female);小鼠(Mice);小鼠, SCID(Mice, SCID);显微镜检查, 共焦(Microscopy, Confocal);模型, 分子(Models, Molecular);磷蛋白类(Phosphoproteins);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质c-akt(Proto-Oncogene Proteins c-akt);重组蛋白质类(Recombinant Proteins);信号传导(Signal Transduction);表面等离激元(Surface Plasmon Resonance)
DOI
10.1158/0008-5472.CAN-08-3839
PMID
19491272
发布时间
2025-05-29
- 浏览16
Cancer research
5073-81页
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