Development of N-[11C]methylamino 4-hydroxy-2(1H)-quinolone derivatives as PET radioligands for the glycine-binding site of NMDA receptors.
作者:
主题词
动物(Animals);放射自显影术(Autoradiography);结合部位(Binding Sites);脑(Brain);甘氨酸(Glycine);小鼠(Mice);分子结构(Molecular Structure);正电子发射断层显像术(Positron-Emission Tomography);蛋白质结合(Protein Binding);喹诺酮类(Quinolones);放射化学(Radiochemistry);放射性药物(Radiopharmaceuticals);受体, N-甲基-D-天冬氨酸(Receptors, N-Methyl-D-Aspartate);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmc.2009.06.014
PMID
19586774
发布时间
2013-11-21
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