Accessing protein methyltransferase and demethylase enzymology using microfluidic capillary electrophoresis.
第一作者:
Tim J,Wigle
第一单位:
Center for Integrative Chemical Biology and Drug Discovery Division of Medicinal Chemistry and Natural Products, Eshelman School of Pharmacy, The University of North Carolina, CB #7363, 120 Mason Farm Road, Chapel Hill, NC 27599-7363, USA.
作者:
主题词
氨基酸序列(Amino Acid Sequence);结合, 竞争性(Binding, Competitive);药物评价, 临床前(Drug Evaluation, Preclinical);电泳, 毛细管(Electrophoresis, Capillary);酶测定(Enzyme Assays);组蛋白脱甲基酶类(Histone Demethylases);组蛋白赖氨酸N-甲基转移酶(Histone-Lysine N-Methyltransferase);动力学(Kinetics);甲基化(Methylation);微流体分析技术(Microfluidic Analytical Techniques);分子序列数据(Molecular Sequence Data);肽类(Peptides);S-腺苷甲硫氨酸(S-Adenosylmethionine);小分子化合物库(Small Molecule Libraries)
DOI
10.1016/j.chembiol.2010.04.014
PMID
20659682
发布时间
2024-06-08
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Chemistry & biology
695-704页
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