Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 2: Discovery of highly potent anti-HIV agents.
第一作者:
Ben,Li
第一单位:
Shanghai Institutes for Biological Sciences, Chinese Academy of Sciences, Shanghai, PR China.
作者:
医学主题词
动物(Animals);抗HIV药(Anti-HIV Agents);CHO细胞(CHO Cells);仓鼠亚科(Cricetinae);仓鼠属(Cricetulus);药物发现(Drug Discovery);吡咯烷类(Pyrrolidines);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2010.05.046
PMID
20674358
发布时间
2014-11-20
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